APG-2449 in Patients With Advanced Solid Tumors

⚠️

This is not medical advice. AI-assisted translation — inaccuracies may occur. Always verify the original and consult your oncologist before taking any steps.

About the trial

APG-2449 is a novel, orally active, multi-targeted tyrosine kinase inhibitor, which inhibits FAK, ALK, and ROS1 with nanomolar potencies. In preclinical studies, APG-2449 demonstrated potent antiproliferative activity in various cancer cell lines as a single agent. In combination treatment, APG-2449 enhanced anti-proliferative activities of several chemotherapeutic and targeted agents. It is indicated that APG-2449 may have a broad therapeutic potential for the treatment of human cancer as a single agent and in combination with other classes of anticancer drugs. APG-2449 is intended for the treatment of patients with advanced solid tumors. Upon completion of the Phase 1 dose escalation study to establish the maximum tolerated dose (MTD), dose-limiting toxicities (DLTs), and/or recommended phase 2 dose (RP2D), several phase Ib/II studies will be implemented accordingly.

Original English text from ClinicalTrials.gov

Who can (and can't) join

✓ Qualifies

  • Rак płuca bez drobnych komórek z mutacją ALK lub ROS1, lub inne zaawansowane nowotwory (przełyk, jajniki, opłucna)
  • Wyniki badań krwi i szpiku kostnego w normie
  • Prawidłowa funkcja nerek i wątroby
  • Prawidłowe funkcjonowanie serca
  • Co najmniej jedna zmiana widoczna na obrazach
  • Oczekiwana długość życia co najmniej 3 miesiące
  • Kobieta w wieku rozrodczym musi mieć ujemny test ciąży
  • Gotowość do stosowania antykoncepcji przez 30 dni po zakończeniu badania

Simplified criteria — AI translation

Trial details

Minimum age
18 Years
Last updated (source)
July 23, 2026
Sex
No restrictions

Therapies / drugs in trial

Locations (9)

Beijing Cancer Hospital

Beijing, China

Fujian Medical University Union Hospital

Fuzhou, China

Fujian Cancer Hospital

Fuzhou, China

Sun-Yat Sen University Cancer Center

Guangzhou, China

The First affiliated hospital, Sun Yat-sen University

Guangzhou, China

Henan Provincial Oncology Hospital

Zhengzhou, China

Union Hospital medical college Huazhong University of Science and Technology

Wuhan, China

Hunan Provincial Oncology Hospital

Changsha, China

Zhejiang Provincial Oncology Hospital

Hangzhou, China

Trial contact

Yifan Zhai, M.D., Ph.D.

Contact information from ClinicalTrials.gov. Contact in English.

Share this trial

Data from ClinicalTrials.gov. AI-assisted translation, last sync: 7/24/2026.

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