RecruitingPhase I/IIEN originalOther cancersMetastatic / advanced

Safety and Tolerability of TNG462 in Patients With MTAP-deleted Solid Tumors

⚠️

This is not medical advice. AI-assisted translation — inaccuracies may occur. Always verify the original and consult your oncologist before taking any steps.

About the trial

This is a first in human study in patients with advanced or metastatic solid tumors known to have an MTAP deletion. The first part of the study is an open-label, dose escalation and the second part is an open label dose expansion in specific MTAP-deleted tumor types. The study drug, TNG462, is a selective PRMT5 inhibitor administered orally. The study is planned to treat up to 225 participants.

Original English text from ClinicalTrials.gov

Who can (and can't) join

✓ Qualifies

  • Wiek co najmniej 18 lat
  • Dobry stan ogólny pacjenta (ECOG 0-1)
  • Potwierdzona diagnoza zaawansowanego lub rozprzestrzenienia się nowotworu
  • Wcześniejsze leczenie standardowe
  • Potwierdzony brak białka MTAP w guzie
  • Prawidłowa funkcja wątroby
  • Prawidłowa funkcja nerek
  • Pisemna zgodę na udział w badaniu

✗ Disqualifies

  • Alergia lub nietolerancja badanego leku lub pembrolizumabu
  • Niekontrolowana choroba towarzysząca utrudniająca udział w badaniu
  • Aktywny zakażenie wymagające leczenia
  • Udział w innym badaniu klinicznym
  • Zaburzenia wchłaniania w przewodzie pokarmowym
  • Aktywny nowotwór w innej lokalizacji
  • Przerzuty do mózgu z objawami neurologicznymi
  • Aktywna choroba wątroby z innego powodu

Simplified criteria — AI translation

Trial details

Minimum age
18 Years
Last updated (source)
April 21, 2026
Sex
No restrictions

Therapies / drugs in trial

Locations (26)

Stanford University

Palo Alto, United States

Grand Valley Oncology

Grand Junction, United States

Florida Cancer Specialists & Research Institute

Lake Mary, United States

Sylvester Comprehensive Cancer Center

Miami, United States

University Chicago Medicine

Chicago, United States

Carle Cancer Center

Urbana, United States

Midwestern Regional Medical Center, City of Hope Chicago

Zion, United States

Massachusetts General Hospital

Boston, United States

Dana Farber Cancer Institute

Boston, United States

Henry Ford Cancer Center

Detroit, United States

New York University Langone Health

New York, United States

Sarah Cannon Tennessee Oncology

Nashville, United States

The University of Texas MD Anderson Cancer Center

Houston, United States

Huntsman Cancer Institute, University of Utah

Salt Lake City, United States

Next Oncology Virginia

Fairfax, United States

CHU de Brest

Brest, France

Centre Berard Leon

Lyon, France

Institut de Cancerologie de l'Ouest - Hôpital Saint Herblain - PPDS

Saint-Herblain, France

Institute Gustav Roussy

Villejuif, France

Vall d'Hebron Barcelona Hospital

Barcelona, Spain

Hospital HM Nou Delfos

Barcelona, Spain

ICO l'Hospitalet - Hospital Duran i Reynals

Barcelona, Spain

Hospital Universitario Fundacion Jimenez Diaz

Madrid, Spain

Hospital de Sanchinarro

Madrid, Spain

Hospital Universitario Virgen de la Victoria

Málaga, Spain

Hospital Universitario Virgen del Rocio

Seville, Spain

Trial contact

Contact information from ClinicalTrials.gov. Contact in English.

Share this trial

Data from ClinicalTrials.gov. AI-assisted translation, last sync: 7/1/2026.

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