A Study to Evaluate the Effect of GDC-4198 Alone and in Combination With Giredestrant Versus Abemaciclib and Giredestrant in Participants With Locally Advanced or Metastatic Estrogen Receptor-Positive (ER+), Human Epidermal Growth Factor Receptor-Negative (HER2-) Breast Cancer

⚠️

This is not medical advice. AI-assisted translation — inaccuracies may occur. Always verify the original and consult your oncologist before taking any steps.

About the trial

The purpose of this study is to assess the safety of GDC-4198 alone and in combination with giredestrant and also the efficacy of GDC-4198 + giredestrant versus abemaciclib + giredestrant in participants with locally advanced or metastatic ER+, HER2- breast cancer. The study consists of 2 phases: Phase Ib and Phase II. Phase Ib will evaluate the safety and pharmacokinetics (PK) of GDC-4198 alone and in combination with giredestrant. Phase II stage will compare the activity and safety of GDC-4198 and giredestrant with abemaciclib and giredestrant.

Original English text from ClinicalTrials.gov

Who can (and can't) join

✓ Qualifies

  • Rak piersi potwierdzony badaniem histologicznym lub cytologicznym, który jest miejscowo zaawansowany lub rozprzestrzeniony (przerzuty).
  • Rak piersi z dodatnimi receptorami estrogenowymi (ER+) i ujemnym receptorem HER2 (HER2-), potwierdzony według wytycznych.
  • Progresja choroby podczas lub po leczeniu innym lekiem (inhibitor CDK4/6) i leczeniem hormonalnym.
  • Choroba, którą można zmierzyć lub ocenić.
  • Ogólny stan zdrowia pacjentki pozwalający na aktywność (grupa 0 lub 1 wg skali ECOG).
  • Przewidywana długość życia co najmniej 6 miesięcy.

✗ Disqualifies

  • Zaawansowane objawy choroby w narządach wewnętrznych, które mogą prowadzić do poważnych powikłań zagrażających życiu w najbliższym czasie.
  • Przeszłość leczenia (poza badaniem) większą niż jedna linia terapii dla choroby zaawansowanej lub z przerzutami.
  • Wcześniejsze chemioterapia w leczeniu raka piersi z przerzutami.
  • Przyjmowanie niektórych leków hormonalnych lub inhibitorów CDK4/6 w ciągu ostatnich 7 lub 21 dni przed rozpoczęciem badania.
  • Problemy z wchłanianiem leków w przewodzie pokarmowym.
  • Inne choroby nowotworowe w ciągu ostatnich 3 lat (z pewnymi wyjątkami).
  • Znane uczulenie na którykolwiek ze składników badanych leków.

Simplified criteria — AI translation

Trial details

Minimum age
18 Years
Last updated (source)
August 10, 2026
Sex
No restrictions

Therapies / drugs in trial

Locations (61)

University of Arizona Cancer Center

Tucson, United States

City of Hope

Duarte, United States

City of Hope - Orange County Lennar Foundation Cancer Center

Irvine, United States

UC San Diego Moores Cancer Center

La Jolla, United States

University of California San Diego Medical Center

San Diego, United States

UCSF Helen Diller Family CCC

San Francisco, United States

Sylvester Comprehensive Cancer Center

Miami, United States

Moffitt Cancer Center

Tampa, United States

Winship Cancer Institute of Emory University

Atlanta, United States

City of Hope® Cancer Center Chicago

Zion, United States

Barbara Ann Karmanos Cancer Institute

Detroit, United States

Maryland Oncology Hematology - Annapolis

Annapolis, United States

Washington University Siteman Cancer Center

St Louis, United States

Rutgers Cancer Institute of New Jersey

New Brunswick, United States

New York Cancer & Blood Specialists

East Patchogue, United States

Montefiore Einstein Cancer Center

The Bronx, United States

Levine Cancer Institute

Charlotte, United States

Novant Health Cancer Institute

Charlotte, United States

Oncology Associates of Oregon, P.C

Eugene, United States

Penn State Health Milton S. Hershey Medical Center

Hershey, United States

University of Pennsylvania - Abramson Cancer Center

Philadelphia, United States

UPMC - Hillman Cancer Center

Pittsburgh, United States

Vanderbilt Breast Center at One Hundred Oaks

Nashville, United States

Texas Oncology (Worth) - USOR

Dallas, United States

University of Utah Huntsman Cancer Institute

Salt Lake City, United States

Virginia Oncology Associates (Norfolk) - USOR

Norfolk, United States

St Vincent's Hospital Sydney

Darlinghurst, Australia

Cancer Research SA

Adelaide, Australia

Hospital do Cancer de Pernambuco - HCP

Recife, Brazil

ONCOSITE Centro de Pesquisa Clínica Em Oncologia

Ijuí, Brazil

Irmandade Da Santa Casa de Misericordia de Porto Alegre

Porto Alegre, Brazil

Hospital de Clinicas de Porto Alegre (HCPA) - PPDS

Porto Alegre, Brazil

Instituto Do Câncer Do Estado de São Paulo Octávio Frias de Oliveira - ICESP

São Paulo, Brazil

Princess Margaret Hospital

Toronto, Canada

Shandong Cancer Hospital

Jinan, China

Fudan University Shanghai Cancer Center - Pudong Campus

Shanghai, China

Tianjin Medical University Cancer Institute & Hospital

Tianjin, China

Institut Jean Godinot

Reims, France

Gustave Roussy

Villejuif, France

Centre Francois Baclesse

Caen, France

Centre Oscar Lambret

Lille, France

Centre Eugene Marquis

Rennes, France

Universitatsklinikum Tubingen

Tübingen, Germany

KEM - Evang. Huyssens-Stiftung Essen-Huttrop

Essen, Germany

Universitatsklinikum Hamburg-Eppendorf

Hamburg, Germany

IRCCS Azienda Ospedaliero Universitaria di Bologna

Bologna, Italy

Istituto Romagnolo per lo Studio dei Tumori Dino Amadori - IRST S.r.l - PPDS

Meldola, Italy

ASST degli Spedali Civili di Brescia - Spedali Civili di Brescia

Brescia, Italy

Ospedale San Raffaele S.r.l. - PPDS

Milan, Italy

Gangnam Severance Hospital, Yonsei University Health System

Seoul, South Korea

Seoul National University Bundang Hospital

Seongnam-si, South Korea

Seoul National University Hospital

Seoul, South Korea

Asan Medical Center.

Seoul, South Korea

Samsung Medical Center

Seoul, South Korea

Severance Hospital, Yonsei University Health System

Seoul, South Korea

The Catholic University of Korea, Seoul St. Mary's Hospital

Seoul, South Korea

Instituto de Investigacion Oncologica Vall dHebron (VHIO) - EPON

Barcelona, Spain

Hospital Beata Maria Ana

Madrid, Spain

Hospital General Universitario Gregorio Maranon

Madrid, Spain

Hospital Universitario 12 de Octubre

Madrid, Spain

Hospital Clinico Universitario de Valencia

Valencia, Spain

Trial contact

Reference Study ID Number: GO46021 https://forpatients.roche.com/ No attachments to email below.

Fastest response: use the inquiry form. https://www.gene.com/contact-us/submit-medical-inquiry

Contact information from ClinicalTrials.gov. Contact in English.

Share this trial

Data from ClinicalTrials.gov. AI-assisted translation, last sync: 7/1/2026.

You can help another person

We fund the Radar, this site, and the development of our Grosz dla Życia fundraising platform from donations and our own resources. Every contribution, even a small one, really helps.